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Publications

Covalent Inhibitors of S100A4 Block the Formation of a Pro-Metastasis Non-Muscle Myosin 2A Complex.

Giroud C. et al, (2024), J Med Chem, 67, 18943 - 18956

Design, Synthesis, and Biological Evaluation of 2-Hydroxy-4-phenylthiophene-3-carbonitrile as PD-L1 Antagonist and Its Comparison to Available Small Molecular PD-L1 Inhibitors.

Ważyńska MA. et al, (2023), J Med Chem, 66, 9577 - 9591

Erratum: Amenamevir by Ugi-4CR (Green Chem. (2023) 25 (1322–1325) DOI: 10.1039/D2GC04869H)

Li X. et al, (2023), Green Chemistry, 25

Discovery and Development Strategies for SARS-CoV-2 NSP3 Macrodomain Inhibitors.

Schuller M. et al, (2023), Pathogens, 12

Amenamevir by Ugi-4CR

Li X. et al, (2023), Green Chemistry

Synthesis of meta-substituted arene bioisosteres from [3.1.1]propellane.

Frank N. et al, (2022), Nature, 611, 721 - 726

Local Anesthetics via Multicomponent Reactions.

Thomaidi M. et al, (2022), ChemMedChem, 17

Supported Gold Nanoparticle-Catalyzed Selective Reduction of Multifunctional, Aromatic Nitro Precursors into Amines and Synthesis of 3,4-Dihydroquinoxalin-2-Ones.

Iordanidou D. et al, (2022), Molecules, 27

Biphenyl Ether Analogs Containing Pomalidomide as Small-Molecule Inhibitors of the Programmed Cell Death-1/Programmed Cell Death-Ligand 1 Interaction

Shaabani S. et al, (2022), Molecules, 27

Synthesis of meta-substituted arene bioisosteres from [3.1.1]propellane

Frank N. et al, (2022)

Author Correction: A phenotypic high-content, high-throughput screen identifies inhibitors of NLRP3 inflammasome activation.

Nizami S. et al, (2021), Sci Rep, 11

A phenotypic high-content, high-throughput screen identifies inhibitors of NLRP3 inflammasome activation.

Nizami S. et al, (2021), Sci Rep, 11

Nanoscale, automated, high throughput synthesis and screening for the accelerated discovery of protein modifiers

Gao K. et al, (2021), RSC Medicinal Chemistry, 12, 809 - 818

Multicomponent reaction-derived covalent inhibitor space

Sutanto F. et al, (2021), Science Advances, 7

Inhibition of the NLRP3 inflammasome by HSP90 inhibitors.

Nizami S. et al, (2021), Immunology, 162, 84 - 91

TEAD-YAP Interaction Inhibitors and MDM2 Binders from DNA-Encoded Indole-Focused Ugi Peptidomimetics.

Kunig VBK. et al, (2020), Angew Chem Int Ed Engl, 59, 20338 - 20342

Multicomponent Reactions: "Kinderleicht"

Neochoritis CG. et al, (2020), Journal of Chemical Education, 97, 3739 - 3745

[18F]Atorvastatin: synthesis of a potential molecular imaging tool for the assessment of statin-related mechanisms of action

Clemente GS. et al, (2020), EJNMMI Research, 10

Late-Stage Copper-Catalyzed Radiofluorination of an Arylboronic Ester Derivative of Atorvastatin.

S Clemente G. et al, (2019), Molecules, 24

Isocyanide-Based Multicomponent Reactions of Free Phenylboronic Acids

Neochoritis CG. et al, (2019), European Journal of Organic Chemistry, 2019, 6132 - 6137

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