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Search results (47)

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Ugi-Tetrazole-Derived α-Aminomethyl Scaffolds Reveal Unexpected Binding Modes in SARS-CoV-2 3CLpro

van der Straat R. et al, (2026), ACS MEDICINAL CHEMISTRY LETTERS

A patent review of peptidylarginine deiminase 4 (PAD4) inhibitors (2014-present).

Aiken SG. et al, (2025), Expert Opin Ther Pat, 35, 611 - 621

Structural Dynamics of the Ubiquitin Specific Protease USP30 in Complex with a Cyanopyrrolidine-Containing Covalent Inhibitor.

O'Brien DP. et al, (2025), J Proteome Res, 24, 479 - 490

Covalent Inhibitors of S100A4 Block the Formation of a Pro-Metastasis Non-Muscle Myosin 2A Complex.

Giroud C. et al, (2024), J Med Chem, 67, 18943 - 18956

Design, Synthesis, and Biological Evaluation of 2-Hydroxy-4-phenylthiophene-3-carbonitrile as PD-L1 Antagonist and Its Comparison to Available Small Molecular PD-L1 Inhibitors.

Ważyńska MA. et al, (2023), J Med Chem, 66, 9577 - 9591

Erratum: Amenamevir by Ugi-4CR (Green Chem. (2023) 25 (1322–1325) DOI: 10.1039/D2GC04869H)

Li X. et al, (2023), Green Chemistry, 25

Discovery and Development Strategies for SARS-CoV-2 NSP3 Macrodomain Inhibitors.

Schuller M. et al, (2023), Pathogens, 12

Amenamevir by Ugi-4CR

Li X. et al, (2023), Green Chemistry, 25, 1322 - 1325

Synthesis of meta-substituted arene bioisosteres from [3.1.1]propellane.

Frank N. et al, (2022), Nature, 611, 721 - 726

Local Anesthetics via Multicomponent Reactions.

Thomaidi M. et al, (2022), ChemMedChem, 17

Supported Gold Nanoparticle-Catalyzed Selective Reduction of Multifunctional, Aromatic Nitro Precursors into Amines and Synthesis of 3,4-Dihydroquinoxalin-2-Ones.

Iordanidou D. et al, (2022), Molecules, 27

Synthesis of meta-substituted arene bioisosteres from [3.1.1]propellane

Frank N. et al, (2022)

Biphenyl Ether Analogs Containing Pomalidomide as Small-Molecule Inhibitors of the Programmed Cell Death-1/Programmed Cell Death-Ligand 1 Interaction.

Shaabani S. et al, (2022), Molecules, 27

Author Correction: A phenotypic high-content, high-throughput screen identifies inhibitors of NLRP3 inflammasome activation.

Nizami S. et al, (2021), Sci Rep, 11

A phenotypic high-content, high-throughput screen identifies inhibitors of NLRP3 inflammasome activation.

Nizami S. et al, (2021), Sci Rep, 11

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