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Search results (12)

« Back to Publications

Crystallographic fragment screening and deep mutational scanning of Zika virus NS2B-NS3 protease enable development of resistance-resilient inhibitors.

Ni X. et al, (2025)

Covalent Inhibitors of S100A4 Block the Formation of a Pro-Metastasis Non-Muscle Myosin 2A Complex.

Giroud C. et al, (2024), J Med Chem, 67, 18943 - 18956

Crystallographic Fragment Screen of Coxsackievirus A16 2A Protease identifies new opportunities for the development of broad-spectrum anti-enterovirals.

Lithgo RM. et al, (2024)

Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3.

Raux B. et al, (2024), Bioorg Med Chem Lett, 98

Turning high-throughput structural biology into predictive inhibitor design.

Saar KL. et al, (2023), Proc Natl Acad Sci U S A, 120

A Chemical Probe for Tudor Domain Protein Spindlin1 to Investigate Chromatin Function.

Fagan V. et al, (2019), J Med Chem, 62, 9008 - 9025

Discovery of a Selective Inhibitor for the YEATS Domains of ENL/AF9.

Christott T. et al, (2019), SLAS Discov, 24, 133 - 141

Development of a YEATS-domain chemical probe

Moustakim M. et al, (2018), ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 256

P2X1 Receptor Antagonists Inhibit HIV-1 Fusion by Blocking Virus-Coreceptor Interactions.

Giroud C. et al, (2015), J Virol, 89, 9368 - 9382

High-Throughput HIV-Cell Fusion Assay for Discovery of Virus Entry Inhibitors.

Marin M. et al, (2015), Assay Drug Dev Technol, 13, 155 - 166

HIV-1-associated PKA acts as a cofactor for genome reverse transcription.

Giroud C. et al, (2013), Retrovirology, 10

Cellular kinases incorporated into HIV-1 particles: passive or active passengers?

Giroud C. et al, (2011), Retrovirology, 8